Bookedited by Norbert Handler and Helmut Buschmann.
Contents:
Introduction. Polypharmacology in Drug Discovery / Oscar Méndez-Lucio, J Jesús Naveja, Hugo Vite-Caritino, Fernando D Prieto-Martínez, José L Medina-Franco
Selectivity of Marketed Drugs. Kinase Inhibitors / Peng Wu, Michael Givskov, Thomas E Nielsen
Repositioning of Drug - New Indications for Marketed Drugs / Ren Kong, Stephen T Wong
Discovery Technologies for Drug Repurposing / Naiem T Issa, Stephen W Byers, Sivanesan Dakshanamurthy
Unselective Drugs in Drug Discovery. Personalized Medicine / Christian Noe, Volker Baumann
Drug Discovery Strategies for the Generation of Multitarget Ligands against Neglected Tropical Diseases / Annachiara Gandini, Federica Prati, Elisa Uliassi, Maria L Bolognesi
Designing Approaches to Multitarget Drugs / Luca Costantino, Daniela Barlocco
The Linker Approach / Daniel Merk, Manfred Schubert-Zsilavecz
Merged Multiple Ligands / Hongming Chen, Udo Bauer, Ola Engkvist
Pharmacophore Generation for Multiple Ligands / Norbert Handler
Cellular Assays / Ye Fang
Therapeutic Areas for Designed Multiple Ligands. Developing Serotonergic Antidepressants Acting on More Than the Serotonin Transporter / Gerard J Marek
Multiple Ligands Targeting the Angiotensin System for Hypertension / Agustin Casimiro-Garcia
Multiple Peroxisome Proliferator-Activated Receptor-Based Ligands / Dmytro Kukhtar, Miquel Mulero, Raul Beltrán-Debón, Cristina Valls, Gerard Pujadas, Santiago Garcia-Vallve
Antibiotics / Jean-Philippe Surivet, Philippe Panchaud
Multiple Ligands in Neurodegenerative Diseases / Julien Lalut, Christophe Rochais, Patrick Dallemagne.